Mgr. Katarína Chalupová, Ph.D.

HANZLOVÁ, Michaela, M. SEDLÁČEK MIŠKEŘÍKOVÁ, A. ROTTEROVÁ, K. CHALUPOVÁ, K. JURKOVÁ, M. HAMŠÍKOVÁ, R. ANDRÝS, A. HALEČKOVÁ, J. SVOBODOVÁ, M. SCHMIDT, O. BENEK, K. MUSÍLEK. Nanomolar Benzothiazole-Based Inhibitors of 17β-HSD10 with Cellular Bioactivity. ACS Medicinal Chemistry Letters. 2023, 14 (12), 1724-1732. ISSN 1948-5875.

OLEKŠÁK, Patrik, M. PSOTKA, M. VANCUROVA, O. SAPEGA, J. BIEBLOVA, M. REINIS, D. RYSANEK, R. MIKYSKOVA, K. CHALUPOVÁ, D. MALIŇÁK, J. SVOBODOVÁ, R. ANDRÝS, H. ŘEHULKOVÁ, V. ŠKOPEK, NL. PHAM, J. BARTEK, Z. HODNY, K. MUSÍLEK. Design, synthesis, and in vitro evaluation of BP-1-102 analogs with modified hydrophobic fragments for STAT3 inhibition. Journal of enzyme inhibition and medicinal chemistry. 2021, 36 (1), 410-424. ISSN 1475-6366.

MEZEIOVA, Eva, M. HRABINOVA, V. HEPNAROVA, D. JUN, J. JANOCKOVA, L. MUCKOVA, L. PRCHAL, Z. KRISTOFIKOVA, T. KUCERA, L. GORECKI, K. CHALUPOVÁ, J. KUNES, J. HROUDOVA, O. SOUKUP, J. KORABECNY. Huprine Y-Tryptophan heterodimers with potential implication to Alzheimer's disease treatment. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2021, 43 (JUL 1), "Article Number: 128100". ISSN 0960-894X.

NEPOVIMOVÁ, Eugenie, L. SVOBODOVA, R. DOLEŽAL, V. HEPNAROVA, L. JUNOVA, D. JUN, J. KORABECNY, T. KUCERA, Z. GAZOVA, K. MOTYKOVA, J. KUBACKOVA, Z. BEDNARIKOVA, J. JANOČKOVÁ, C. JESUS, L. CORTES, J. PINA, D. ROSTOHAR, C. SERPA, O. SOUKUP, L. AITKEN, R. HUGHES, K. MUSÍLEK, L. MUCKOVA, P. JOST, M. CHVOJKOVA, K. VALES, M. VALIS, Ž. CHRIENOVÁ, K. CHALUPOVÁ, K. KUČA. Tacrine – Benzothiazoles: Novel class of potential multitarget anti-Alzheimeŕs drugs dealing with cholinergic, amyloid and mitochondrial systems. Bioorganic Chemistry. 2021, 107 (February), "Article number 104596". ISSN 0045-2068.

MEZEIOVA, Eva, K. CHALUPOVÁ, E. NEPOVIMOVÁ, L. GORECKI, L. PRCHAL, D. MALIŇÁK, K. KUČA, O. SOUKUP, J. KORABECNY. Donepezil Derivatives Targeting Amyloid-beta Cascade in Alzheimer's Disease. Current Alzheimer research. 2019, 16 (9), 772-800. ISSN 1567-2050.

CHALUPOVÁ, Katarína, J. KORABECNY, M. BARTOLINI, B. MONTI, D. LAMBA, R. CALIANDRO, A. PESARESI, X. BRAZZOLOTTO, A. GASTELLIER, F. NACHON, J. PEJCHAL, M. JAROSOVA, V. HEPNAROVA, D. JUN, M. HRABINOVA, R. DOLEŽAL, JZ. KARASOVA, M. MZIK, Z. KRISTOFIKOVA, J. MISIK, L. MUCKOVA, P. JOST, O. SOUKUP, M. BENKOVA, V. SETNICKA, L. HABARTOVA, M. CHVOJKOVA, L. KLETECKOVA, K. VALES, E. MEZEIOVA, E. ULIASSI, M. VALIS, E. NEPOVIMOVÁ, ML. BOLOGNESI, K. KUČA. Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease. European journal of medicinal chemistry. 2019, 168 (April), 491-514. ISSN 0223-5234.

MZIK, M., J. ZD'AROVA-KARASOVA, K. CHALUPOVÁ, J. KORABECNY, V. PALICKA, V. SESTAK. UHPLC-HRMS study of anti-Alzheimer's drug candidates: metabolism of 7-MEOTA-tryptophan hybrids hampers their passage into brain. Journal of pharmaceutical and biomedical analysis. 2019, 174 (září), 134-144. ISSN 0731-7085.

MEZEIOVA, Eva, K. ŠPILOVSKÁ, E. NEPOVIMOVÁ, L. GORECKI, O. SOUKUP, R. DOLEZAL, D. MALIŇÁK, J. JANOCKOVA, D. JUN, K. KUČA, J. KORABECNY. Profiling donepezil template into multipotent hybrids with antioxidant properties. Journal of enzyme inhibition and medicinal chemistry. 2018, 33 (1), 583-606. ISSN 1475-6366.